I-Andarine iyi-SARM enemiphumela emihle kakhulu ye-androgenic njengoba izungeze i-33% yamandla e-testosterone lapho inamathisela ku-AR.I-Andarine iphinde ikhulise inani lesisindo somzimba esikhiqizwa ngokususa i-AR ku-testosterone yemvelo yomuntu ukuze ibe nomthelela onamandla.
I-Andarine iyi-SARM eguquguquka kakhulu eyake yadalwa.Akukhona nje kuphela ukuthi i-SARM yokuqala evunyelwe isifundo socwaningo lwesiteji se-2, isibe yi-SARM ehlaziywe kakhulu futhi ephenywa kuze kube manje.Ngemva kokutholakala kwamandla ayo e-anabolic, inhloso eyinhloko ye-Andarine ihlose ukuthuthukisa enye indlela yokwelapha ukuchithwa kwemisipha ehlobene neminyaka, i-osteoporosis, kanye nezimpawu ezifanayo ze-hypogonadism, noma isifo sezinso sokuphela.
Ngaphandle kokugcina isisindo somzimba omncane, i-Andarine ingasiza futhi ukuyithuthukisa.Kusukela esifundweni se-1, i-Andarine inikeze ubufakazi bokukhuphuka kwe-3.3 lbs ezinsukwini ezingaphansi kwezingu-90 ngaphandle kokwenyuka kokuzivocavoca noma ushintsho ekudleni kwansuku zonke.Umphumela ongahlosiwe (noma uzuze uma uthanda) ukwehla kwamafutha omzimba.Ukuncipha kwamafutha omzimba kuncike kufuzo lomuntu, kodwa kuzoba nemiphumela eqinile emandleni omzimba okukhipha izicubu ezinamafutha.I-Andarine itholwe ingenakho ukuhlobana okuhle kuphela (amandla ekubophezeleni kuma-androgen receptors), kuyilapho futhi yethula imiphumela emikhulu ye-anabolic kunezinye i-steroids yendabuko.
Ngaphandle kwezinzuzo zayo zokwakha imisipha, i-Andarine ngeke ibangele ukulimala kwesibindi, ingavimbela i-gynecomastia (amabele akhulisiwe emadodeni) futhi ingasiza ekuthuthukiseni impilo yakho yonke.
I-Andarine (GTx-007, S-4) iyisiguquli se-androgen receptor (SARM) esikhethiwe sophenyo esakhiwe yi-GTX, Inc ukuze kulashwe izimo ezifana nokuwohloka kwemisipha, i-osteoporosis kanye ne-benign prostatic hypertrophy, kusetshenziswa i-bicalutamide engeyona i-steroidal androgen njenge- inhlanganisela yokuhola.
I-Andarine iyi-agonist eyingxenye yomlomo esebenzayo ye-androgen receptors.Inamandla amancane kokubili kwe-anabolic kanye nemiphumela ye-androgenic kunamanye ama-SARM.Kumodeli wezilwane we-benign prostatic hypertrophy, i-andarine yaboniswa ukunciphisa isisindo se-prostate ngokusebenza okufanayo kwe-finasteride, kodwa ngaphandle kokukhiqiza. noma yikuphi ukuncipha kwesisindo somzimba noma imiphumela engemihle ephikisana ne-androgenic.[3]Lokhu kuphakamisa ukuthi iyakwazi ukuvimba ngokuncintisana ukubophezela kwe-dihydrotestosterone ekuhlosweni kwayo kwe-receptor ku-prostate gland, kodwa imiphumela yayo ye-agonist ingxenye kuma-androgen receptors ivimbela imiphumela engathandeki ehambisana nezidakamizwa ezilwa ne-androgenic ngokuvamile ezisetshenziselwa ukwelashwa kwe-BPH.

Imiphumela ye-Andarine (S4) ingasukela ekubhujisweni kuya ekusikeni nasekuguqulweni komzimba okuphelele;Nokho, ukunqwabelana (ukuzuza kwemisipha/ubuningi) kuzoba buthaka kakhulu ezindaweni ezintathu.I-S4 ayaziwa ngokupakisha ezicutshini eziningi ezithambile, kodwa ukuzuza okunciphile kungenziwa futhi kufanele kwenziwe ukuhlinzeka ngama-calories anele akhona kanye nokukhuthazwa kwemisipha (ukuzivocavoca umzimba).Kumsubathi wangaphandle kwesizini ofuna ukupakisha ngokwesayizi ngempela, lona akuwona umkhiqizo abazofuna ukusekela uhlelo lwabo nxazonke nakuba kungaba isengezo esiqinile ohlelweni, hhayi into ezimele.I-Andarine yaziwa kakhulu ngokusiza ekwandeni kwamandla.Ukwandisa amandla kungaba inzuzo uma uzama ukukhula njengoba kuvumela umuntu ukuba aphakamise izinsimbi ezinzima.Nokho, amandla nosayizi akuhambisani ngaso sonke isikhathi futhi akukwazi ukusetshenziswa njengegeji lapho uzama ukukhula.Kungenzeka kakhulu ukuzuza isisindo esincane noma esingenalutho futhi ukhulise amandla naphezu kokungakhushulwa kosayizi.
Ukusika kuzoba lapho i-Andarine (S4) igqama ngempela futhi ngenxa yezizathu ezimbalwa.Inhloso eyinhloko yanoma yiluphi uhlelo lokusika ukulahlekelwa amafutha omzimba.Ukuze umuntu alahlekelwe amafutha emzimbeni kufanele ashise ama- kilojoule amaningi kunalawo awadlayo, okuzobeka izicubu zezicubu ezithambile engozini.I-S4 supplementation inganikeza izindlela zokuvikela izicubu zemisipha ngesikhathi sokuntuleka kwekhalori.Uma izicubu zilondolozwa, i-metabolism izoqhubeka nokuvutha ngamandla.Uma izicubu zilahlekile, i-metabolism inganciphisa ukwenza ukulahlekelwa kwamafutha kube nzima kakhulu.Enye idatha iphinde ibonise i-S4 ukuze ikhulise ngokuqondile i-lipolysis (ukulahlekelwa kwamafutha) nakuba kungacaci ukuthi lokhu kuthinta kubaluleke kangakanani.Ngokulinganayo kunenzuzo ohlelweni lokusika, i-Andarine iboniswe ukwandisa ubulukhuni nencazelo ngokuphawulekayo emzimbeni obuthakathaka.Ukuqina kanye nemiphumela yamandla yale SARM ivame ukufaniswa ne-anabolic steroid Winstrol.Njengebhonasi eyengeziwe, ngezici ezikhulayo zamandla e-S4, kuyilapho amandla angase angakhuli lapho usika, uma usebenzisa le SARM ungase uthole kahle ukuthi ugcina amandla akho amaningi abeyobe enciphile.
Kumuntu othanda ukuqina wansuku zonke, lokhu kungase kube enye yama-SARM angcono kakhulu emakethe.Akwenzeki ukuzuza inani elikhulu lomsipha bese uhlakazeka nganoma yimuphi umkhiqizo.Uma ufuna ukuya ngokwedlulele kunoma iyiphi indlela, kufanele ukhethe isiqondiso esisodwa ngesikhathi.Kodwa uma ufuna uguquko oluningi, hhayi ukwanda okukhulu kosayizi noma ukuklebhula ethanjeni kodwa ukubukeka komzimba ogwini nokwanda kokusebenza kwezemidlalo, lokhu kungenye ye-SARM engcono etholakalayo.Ngenxa yomphumela ongemuhle wemvelo enobungane, futhi ingenye ekhanga kakhulu.
I-S-4 kufanele ithathwe ku-50mg-75mg, izinsuku ezingu-5 ngaphandle kwesonto, amaviki angu-12-16.Njengoba kushiwo ngaphambili, i-S-4 ayidingi ukuthathwa ngezikhathi ezi-3 ezihlukene usuku lonke;kodwa kubantu abakhetha le ndlela, umthamo we-25mg (cishe uhhafu wemililitha) unconywa kanye nokudla kwakho kokuthathu okuyinhloko.
Nakulokhu, njengoba kushiwo ngenhla, i-S-4 inalo iphuzu lokunciphisa ukubuyisela.Lokhu kusho ukuthi ukusetshenziswa kwe-S-4 kudlule i-75mg noma ukusetshenziswa kwe-S-4 ngaphezu kwamaviki e-16 ngeke kubangele noma yikuphi ukungezwa kwemisipha eyengeziwe.Ngeke kube nokwenyuka kwemiphumela engemihle, kodwa uzobe usebenzisa ingcuphe yokungazweli kwe-AR futhi umoshe umkhiqizo wakho nakanjani.Ukuphuza nge-S-4 isikhathi esingaphansi kwamaviki angu-6-8 akunconywa futhi ngeke kuvumele umcwaningi ukuthi abonele izinzuzo ezigcwele zomkhiqizo.
Umthamo onconyiwe wokusika ngu-50 mg wamaviki angama-6-8.Kufanele uyisebenzise nsuku zonke bese uthatha izinsuku ezi-2 zokuphumula.Ukuthatha i-S4 nsuku zonke ubude bomjikelezo kungaholela ekushintsheni kwamehlo.
* Sinendlela ekhethekile yokungakwazi ukuthumela amagremu angu-50 kuya kumikhiqizo engu-50kg ngesikhathi.
* Singanikela ngempushana encibilikayo ibe yisevisi ye-liquid.Futhi sithumele uketshezi emabhodleleni akhethekile.
* Ngokwesicelo sakho kanye nenani lokuthengayo, sinezindlela ezimbalwa zokupakisha ozikhethele zona.ukuphepha nokuthunyelwa okusheshayo kuwe.
* Ithimba lokupakisha eliqeqeshwe kahle neliqeqeshekile.
* Izithombe zokupakisha kanye nekhodi yokupakisha kunikezwa kungakapheli amahora ayi-12 ngemuva kokuthola inkokhelo
* Isevisi enhle kakhulu ngemuva kokuthengisa
* Sihlinzeka ngenqubomgomo yokuthunyelwa kabusha Kwanoma yimiphi imibuzo noma izinkinga ngemva kokuthola umkhiqizo, sicela ukhululeke ukuxhumana nathi.Izinkinga bezizoxazululwa ngokushesha

Into yokuhlola | Ukuhlaziya Ukucaciswa | Umphumela |
Incazelo | i-crystalline powder | Kuyavumelana |
Ibanga lokuncibilika | 129°C~132°C | 130.8°C-131°C |
Ukulahlekelwa ekomisweni | ≤0.5% | 0.20% |
Ukuzungezisa okuqondile | -58°~-62°(C=1,ku-CH3OH) | -61.05° |
Umlotha one-sulphate | ≤0.1% | 0.08% |
Izinsimbi ezinzima | ≤10ppm | Kuyavumelana |
Ama-Chloride | ≤0.02% | Kuyavumelana |
Ama-sulfate | ≤0.02% | Kuyavumelana |
I-Fluorine | 14.7%~17.9% | 15.2% |
I-solvent eyinsalela | I-Methanol ≤0.2% I-Isopropanol ≤0.2% I-Ethyl acetate≤0.2% I-Chloroform ≤0.2% | 0.0% 0.0% 0.0% 0.0% |
Izinto ezihlobene (HPLC) | Ukungcola okukodwa ≤0.2% Ukungcola okuphelele ≤0.5% | 0.05% 0.08% |
Isivivinyo | ≥99.5% | 99.9% |
Isiphetho | Ngokuvumelana nereferensi |
Ukusika (ukusetshenziswa okungcono kakhulu kwe-S4) |
|
Okokubuyisela |
|
Ukuze Uzuze Imisipha Eqinile namandla (ngaphandle kokuqunjelwa) |
|
I-Hjtc (Xiamen) Industry Co., Ltd. Ingumhlinzeki wohlobo olusha ochwepheshile we-Pharmaceutical Packaginga &Steroids Raw Materials .Ifekthri itholakala esifundazweni sase-hubei.Inkampani yethu yajabulela idumela elihle ekhaya naphesheya kwezilwandle ngaphansi kwenkolelo "yokuphathwa kobuqotho, ukulawulwa kwekhwalithi kanye nokuma kweKhasimende".Umkhiqizo wenkampani oncintisanayo ngu I-Pharmaceutical Raw Materials and intermediates, Eminyakeni yamuva, inkampani yenze impumelelo enkulu kuma-steroids powder eluhlaza.umkhiqizo wethu ulingana namazinga e-ISO9001 kanye ne-ISO2000 kazwelonke futhi ngokuvamile sithunyelwa eNyakatho naseNingizimu Melika, eYurophu, eMpumalanga Ephakathi, e-Asia Pacific kanye Indawo yase-Afrika, ukuze kusungulwe ubudlelwano bokubambisana besikhathi eside nobuzinzile namakhasimende emhlabeni.


Igama Lomkhiqizo | Inombolo ye-CAS. | Igama Lomkhiqizo | Inombolo ye-CAS. |
Sarms | |||
Ostarine / MK-2866 | 841205-47-8 | I-MK-677 | 159752-10-0 |
I-Cardarine / GW-501516 | 317318-70-0 | I-Andarine / S4 | 401900-40-1 |
I-Ligandrol / LGD-4033 | 1165910-22-4 | I-RAD140 | 118237-47-0 |
I-SR9009 | 1379686-30-2 | I-SR9011 | 1379686-29-9 |
YK11 | 431579-34-9 | GW0742 | 317318-84-6 |
Lapha | 2627-69-2 | S-23 | 1010396-29-8 |
I-PRL-8-53 | 51352-87-5 | RU58841 | 1270138-41-4 |
I-NSI-189 | 1270138-40-3 | I-ACP105 | 899821-23-9 |
I-NSI-189 i-phosphate | 1270138-41-4 | AC 262536 | 870888-46-3 |
I-Nootropic | |||
I-Sunifiram | 314728-85-3 | I-Coluracetam | 135463-81-9 |
I-Fasoracetam | 110958-19-5 | I-Noopept | 157115-85-0 |
Adrafinils | 63547-13-7 | I-Unifiram | 272786-64-8 |
I-Carphedon | 77472-70-9 | I-Pramiracetam | 68497-62-1 |
I-Anesthetic / Pain Killer | |||
Isisekelo se-Tetracaine | 94-24-6 | I-Prilocaine hydrochloride | 1786-81-8 |
I-Tetracaine hydrochloride | 136-47-0 | I-Proparacaine hydrochloride | 5875-06-9 |
I-Lidocaine hydrochloride | 73-78-9 | I-Pramoxine hydrochloride | 637-58-1 |
I-Linocaine Base | 137-58-6 | I-Procainamide hydrochloride | 614-39-1 |
I-benzocaine hydrochloride | 23239-88-5 | I-Ropivacaine hydrochloride | 98717-15-8 |
I-Benzocaine Base | 94-09-7 | I-Articaine hydrochloride | 23964-57-0 |
I-Procaine | 59-46-1 | I-Bupivacaine | 2180-92-9 |
I-Procaine hydrochloride | 1951/5/8 | I-Mepivacaine hydrochloride/Carbocaine | 1722-62-9 |
I-Prilocaine | 721-50-6 | i-dibucaine hydrochloride | 61-12-1 |
Okunye Okuphakathi Kwemithi | |||
I-Flibanserin/Bimt 17/ | 167933-07-5 | I-Flibanserin HCl | 147359-76-0 |
7,8-dihydroxyflavones / 7,8-DHF | 38183-03-8 | 4'-Dimethylamino 7,8-Dihydroxyflavone | 1205548-00-0 |
1-Chloro-3,5-di-O-toluoyl-2-deoxy-D-ribofuranose | 3601-89-6 | P1301 | 1345680-97-8 |
I-Trikiribine | 35943-35-2 | 2,3-dichloroquinoxaline | 2213-63-0 |
2-Chloropropiophenone | 6084-17-9 | I-Pirespa | 53179-13-8 |
I-MGF | 2mg/ibhodlela |
5mg/ibhodlela | |
I-PEG-MGF | 2mg/ibhodlela |
I-CJC-1295 ene-DAC | 2mg/ibhodlela |
I-CJC-1295 ngaphandle kwe-DAC | 2mg/ibhodlela |
I-PT141 | 10mg/ibhodlela |
MT-1 | 10mg/ibhodlela |
MT-2 | 10mg/ibhodlela |
I-GHRP-2 | 5mg/ibhodlela |
10mg/ibhodlela | |
I-GHRP-6 | 5mg/ibhodlela |
10mg/ibhodlela | |
I-Ipamorelin | 2mg/ibhodlela |
5mg/ibhodlela | |
I-Hexarelin | 2mg/ibhodlela |
I-Sermorelin | 2mg/ibhodlela |
I-Oxytocin | 2mg/ibhodlela |
TB500 | 2mg/ibhodlela |
5mg/ibhodlela | |
I-Pentadecapeptide BPC 157 | 2mg/ibhodlela |
Isiqephu esingu-176-191 | 2mg/ibhodlela |
5mg/ibhodlela | |
I-Triptorelin | 2mg/ibhodlela |
I-Tesamorelin | 2mg/ibhodlela |
I-Gonadorelin | 2mg/ibhodlela |
10mg/ibhodlela | |
I-DSIP | 2mg/ibhodlela |
Selank | 5mg/ibhodlela |
I-IGF-1LR3 | 0.1mg / ibhodlela |
1mg/ibhodlela | |
I-ACE 031 | 1mg / vial (95%) |
1mg / vial (85%) | |
I-GDF-8 | 1mg / vial (95%) |
1mg / vial (85%) |
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