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I-Fareston (i-Toremifene Citrate) ivimbela i-hormone ye-estrogen ekubopheni.
I-Fareston iyi-Selective Estrogen Receptor Modulator (SERM) futhi ingenye ye-SERM entsha emakethe.I-Fareston yaqala ukuthola imvume ye-FDA ngo-1997 nge-GTx INC. futhi ikhiqizwa emazweni amaningi emhlabeni jikelele.I-compound ifana kakhulu ne-Nolvadex (Tamo...Funda kabanzi -
Vardenafil ukuze i-erection itholakale noma igcinwe.
I-Levitra iyimithi ethandwayo ye-erectile dysfunction (ED) yekilasi lemithi ye-phosphodiesterase 5 inhibitor (PED5).I-Bayer, i-GlaxoSmithKline kanye ne-Schering-Plough bathuthukise umuthi we-ED, kodwa kusukela ngo-2005 i-Bayer igcine amalungelo aphelele.I-Levitra ifana kakhulu ne-pop...Funda kabanzi -
Umsebenzi we-Viagra ulula uma kuqhathaniswa - ikhulula imisipha futhi ikhulise ukugeleza kwegazi epipini.
I-Sildenafil, evame ukubizwa ngegama lokuhweba i-Viagra imithi yomlomo esetshenziselwa ukwelashwa kwe-erectile dysfunction (ED).I-Pfizer ikhishwe ngokuthengisa i-Viagra ngo-1996 iyenza ngokusemthethweni isidakamizwa sokuqala esake savunyelwa yi-FDA sokwelashwa kwe-ED.Kuze kube yimanje...Funda kabanzi -
I-Cialis izokhiqiza ama-erections amahora we-36-48 kusuka kumthamo owodwa lapho i-Viagra inqunyelwe emahoreni angu-4-6 kusuka kumthamo owodwa owodwa.
I-Tadalafil ingenye yemithi ethandwa kakhulu emakethe ye-erectile dysfunction (ED) futhi ivame ukuhlotshaniswa negama lomkhiqizo i-Cialis.Ikhishwe yi-GlaxoSmithKline ngo-2003 futhi manje ephethwe ngu-Eli Lilly, i-Cialis ifana kakhulu nomuthi odumile we-ED Viagra...Funda kabanzi -
I-Aromasin inamandla okuvimba i-aromatization, ebuye ivimbele ukukhiqizwa kwe-estrogen, futhi ngaleyo ndlela yehlise amazinga e-serum estrogen emzimbeni.
I-Exemestane iyi-steroidal Aromatase Inhibitor (AI) eyaziwa kakhulu ngokuthi i-Aromasin.Eqinisweni, igama lomkhiqizo we-Aromasin ukuphela kohlobo lwebanga lezemithi lwe-Exemestane AI ngenxa yelungelo lobunikazi eliqinile u-Upjohn aligcinile emkhiqizweni.Ngenkathi ilawulwa ngokuqinile...Funda kabanzi -
Kumsebenzisi we-anabolic steroid, imiphumela ye-Arimidex (Anastrozole) iyaziswa kakhulu emandleni ayo okuvikela ngokumelene nemiphumela emibi ehlobene ne-estrogenic.
Imisebenzi Nezici ze-Arimidex: Imisebenzi nezici ze-Arimidex nakuba zinamandla zilula kakhulu.Njenge-AI i-Arimidex isebenza ngokuvimbela i-enzyme ye-aromatase, ebhekene nokukhiqizwa kwe-estrogen.Ngokuvimbela inqubo ye-aromatase, i-A...Funda kabanzi -
Imiphumela yokuthuthukiswa kwe-IPT-141 kusifiso socansi (i-libido), ukuthuthukiswa kokwaneliseka ngokocansi (futhi kuhlobene ne-libido) kanye nokungasebenzi kahle kwe-erectile.
I-IPT-141, ngezinye izikhathi ebizwa ngokuthi i-PT-141 futhi kamuva nje ngaphansi kwegama elithi Bremelanotide iyi-hormone ye-peptide etholakala ku-Melanotan II.I-Melanotan II (MT2) yathuthukiswa ngenhloso yokugqugquzela ukushukwa kwesikhumba, kodwa kwatholakala ngaphezu kuka-90% wazo zonke izifundo ngesikhathi sokuhlolwa...Funda kabanzi -
I-CJC-1295 iyihomoni ye-peptide elingisa amakhono nemiphumela ye-GHRH, ihomoni eyenzeka ngokwemvelo emzimbeni womuntu.
I-CJC-1295 iyihomoni ye-peptide eyakhiwe yi-ConjuChem Biotechnologies esebenza njenge-Growth Hormone Releasing hormone noma i-GHRH.I-GHRH ihomoni enesibopho sokugqugquzela ukukhishwa kweHormone Yokukhula Komuntu (HGH).Ngamagama alula, singase sithi i-GHRH ise-pitu...Funda kabanzi -
Imiphumela yeCardarine (GW-501516) isiza kakhulu ngokulahlekelwa kwamafutha.
I-GW-501516, eyaziwa kangcono ngokuthi i-Cardarine, umuthi oyingqayizivele ohlukaniswa ngokusemthethweni njenge-PPAR receptor agonist (PPAR-RA).Ucwaningo lwalo muthi lwaqala ngo-1992 emzamweni ohlangene phakathi kwe-GlaxoSmithKline (GSK) kanye ne-Ligand Pharmaceuticals.Ucwaningo ngalo mkhiqizo ...Funda kabanzi -
Abasubathi be-LGD4033 Off-season noma i-bulking bangalindela ukuthola amandla abalulekile kanye nesisindo somzimba ngamakhalori anele.
I-LGD-4033, eyaziwa kangcono ngokuthi i-Anabolicum i-Selective Androgen Receptor Modulator (SARM) efana ne-testosterone i-anabolic kodwa ngaphandle kwemiphumela ebonisa ngokuphawulekayo ngaphandle kwezicubu zemisipha.I-Ligand Pharmaceuticals, i-ligand, ibhekisela kuma-molecule asebenzayo, ...Funda kabanzi -
I-TB-500 ingasetshenziswa ukwelapha izinyembezi zemisipha noma ubunzima, ukuvuvukala kwemisipha kanye nokulimala kwesikhumba.
I-TB-500 iyi-hormone ye-peptide fragment esetshenziswa ngokuyinhloko ekwelapheni ukulimala okuhlukahlukene kwemisipha noma ubuhlungu obubangelwa ukuvuvukala.Incane kakhulu idatha yomuntu esemthethweni etholakalayo yalo mkhiqizo;kodwa-ke, bekuyi-hormone yesikhathi eside esetshenziswa kumahhashi omjaho.I-TB-500...Funda kabanzi -
I-Sermorelin inqunyelwe ngokuyinhloko izingane ezingakhiqizi i-GH ngendlela efanele futhi zihluleka ukukhula ngendlela enempilo ngenxa yalokho.
I-Sermorelin acetate iyi-analogue ye-peptide esanda kuhlanganiswa (eyenziwe ngumuntu) ye-hormone yokukhula ekhulula i-hormone (GHRH) i-hormone eyenzeka ngokwemvelo ekhiqizwa ku-hypothalamus futhi ikhuthaze futhi ilawule ukukhiqizwa kwe-hormone yokukhula (GH) ngaphakathi kwe-pituitary g...Funda kabanzi